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BX795 Inhibitor

InhA, Func 702675-74-9
Catalog No. ABIN3220297
$161.00
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  • Application
    Inhibition Assay (InhA), Functional Studies (Func)
    Purpose
    BX795 is a potent and specific PDK1 inhibitor with IC50 of 6 nM, 140- and 1600-fold more selective for PDK1 than PKA and PKC in cell-free assays, respectively. Meanwhile, in comparison to GSK3β more than 100-fold selectivity observed for PDK1.
    Characteristics
    Target: PDK inhibitor,c-Kit inhibitor, CDK inhibitor, PKA inhibitor
    Receptor: PDE1/TBK1,c-kit,CDK2,PKA
    Purification
    All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
    Purity
    98 %
    Formula
    C23H26IN7O2S
    Solubility
    DMSO > 100mM
  • Background
    Cell Cycle/Checkpoint,PI3K/Akt/mTOR Signaling,Tyrosine Kinase/Adaptors
    Molecular Weight
    591.47 g/mol
    CAS-No
    702675-74-9
  • Application Notes
    Optimal working dilution should be determined by the investigator.
    Restrictions
    For Research Use only
  • Format
    Solid
    Storage
    -20 °C
    Storage Comment
    For the majority of compounds, they could be dissolved in DMSO or other organic solvent.
    Their stock solution can be stored at -20°C for up to 3 months and aliquoted for sampling convenience.
    Several freeze/thaw cycles should not damage the activity of our small molecule products.
    However, in many instances the aqueous solutions of some compounds need to be made fresh and cannot be stored. For these compounds, their solution should be prepared just before use and stored no longer than 24 hours.
    Expiry Date
    24 months
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