Defactinib (VS-6063, PF-04554878)

Details for Product No. ABIN3220511
Application
Inhibition Assay (InhA), Functional Studies (Func)
Options
Purpose Defactinib (VS-6063, PF-04554878) is a selective, and orally active FAK inhibitor. Phase 2.
Characteristics Tradename: PF-04554878, VS-6063
Target: FAK inhibitor
Receptor: FAK
Purification All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
Purity 98 %
Formula C20H21F3N8O3S
Solubility 10 mM in DMSO
Background Angiogenesis
Molecular Weight 510.49 g/mol
CAS-No 1073154-85-4
Application Notes Optimal working dilution should be determined by the investigator.
Restrictions For Research Use only
Format Solid
Storage -20 °C
Storage Comment For the majority of compounds, they could be dissolved in DMSO or other organic solvent.
Their stock solution can be stored at -20°C for up to 3 months and aliquoted for sampling convenience.
Several freeze/thaw cycles should not damage the activity of our small molecule products.
However, in many instances the aqueous solutions of some compounds need to be made fresh and cannot be stored. For these compounds, their solution should be prepared just before use and stored no longer than 24 hours.
Expiry Date 24 months